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Updated: Jan 29 2019

Immunosuppressants

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https://upload.medbullets.com/topic/120715/images/5212017mdstep1immunotargetsofimmunosuppressants.jpg
  • Snapshot
    • A 40-year-old woman presents to the emergency department with worsening lower extremity weakness and decreased visual acuity of the right eye. She reports that her symptoms progressively worsened over the course of a week and after developing a urinary tract infection. Medical history is significant for multiple sclerosis treated with rituximab. Physical examination is significant for 1/5 strength in the lower extremities and an afferent pupillary defect appreciated in the right eye. Magnetic resonance imaging of the brain and spine shows new hyperintense lesions. She is started on intravenous methylprednisolone.
  • Immunosuppressants
    • Immunosuppressants
      Medication
      Clinical Use
      Mechanism of ActionAdverse Effects
      Cyclosporine
      • Rheumatoid arthritis
      • Psoriasis
      • Transplant rejection prophylaxis
      • Calcineurin inhibitor impairs
        • IL-2 production and release
        • IL-2-induced T-cell activation
      • Nephrotoxicity
      • Neurotoxicity
      • Hirsutism
      • Gingival hyperplasia
      • Hypertension
      • Hyperlipidemia
      Tacrolimus (FK506)
      • Transplant rejection prophylaxis
      • Calcineurin inhibitor via binding with intracellularFKBP-12protein which impairs
        • IL-2 production and release
        • IL-2-induced T-cell activation
      • Nephrotoxicity
      • Neurotoxicity
      • ↑ risk of diabetes
      Sirolimus (Rapamycin)
      • Lymphangioleiomyomatosis
      • Renal transplantation prophylaxis
      • mTOR inhibitor via binding with intracellularFKBP-12 protein which
        • ↓ cytokine-induced T-cell proliferation
      • Pancytopenia
      • Hyperlipidemia
      • Edema
      • Insulin resistance
      Basiliximab
      • Renal transplantation prophylaxis
      • Targets the α-chain of the IL-2 receptor complex which is expressed on activated T-cells
      • Edema
      • Tremor
      • Hypertension
      Azathioprine
      • Rheumatoid arthritis
      • Renal transplantation
      • Inflammatory bowel disease
      • Aprecursor of 6-mecaptopurine which
        • incorporates itself into the cell's DNA and halts replication
      • Pancytopenia
      • Hepatotoxicity
      Mycophenolate mofetil
      • Organ transplantation
      • Lupus nephritis
      • Inosine monophosphate dehydrogenase (IMPDH) inhibitor which
        • impairs guanosine nucleotide synthesis
      • Gastrointestinal upset
      • Pancytopenia
      • Hypertension
      • Hyperglycemia
      Corticosteroids
      • A number of autoimmune and inflammatory disorders
      • NF-κB inhibitor
      • Induces T-cell apoptosis
      • Hyperglycemia
      • Osteoporosis
      • Cushing syndrome
      • Adrenocortical atrophy
      • Peptic ulcers
      • Cataracts
      • Avascular necrosis
      • Psychosis
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